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CDRH3 conformational rigidity reduces cross reactivity

CDRH3 conformational rigidity reduces cross reactivity

Created Sep 19, 2024Modified Apr 21, 2026

  • cdrh3
  • antibody-developability/polyspecificity
  • antibody-antigen-interactions/misc

Summary

Conformational rigidity in CDRH3 reduces polyreactivity (1).

See also

  • Conformational entropy in antibodies is inversely proportional to antigen affinity
  • CDR3 loops encode specificity while CDR1 and CDR2 encode cross-reactivity
1.
Fernández-Quintero ML, Loeffler JR, Bacher LM, Waibl F, Seidler CA, Liedl KR. Local and Global Rigidification Upon Antibody Affinity Maturation. Frontiers in Molecular Biosciences. 2020;7. Available from: https://doi.org/10.3389/fmolb.2020.00182

Graph View

Backlinks

  • Antibody-antigen binding modes are not necessarily defined by induced fit
  • Arginine residues in CDRH3 increases promiscuity

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